BRD3-2 Bromodomain Assay Service (AlphaScreen)

BRD3-2-His Reader Domain Assay for compound screening and profiling using the AlphaScreen assay format to measure compound binding to the target.

Target Overview
CAT#

BRD3-2

Enzyme

Human BRD3-2

Synonyms

Bromodomain-containing protein 3 domain 2, RING3-like protein, KIAA0043, RING3L

Substrates

Histone H4 peptide (1-21) K5/8/12/16Ac

Assay Properties
Reaction

AlphaScreen Binding assay

Readout

Fluorescence

Reference Compound IC50s
Compounds IC50 (nM)
JQ-1 25
PFI-1 170
Scientific Information

Q15059 (http://www.uniprot.org/uniprot/Q15059)

Screening Location

Malvern, USA

Further information

More information can be found on our website Reader Domain Assay Services.

Reference Compound IC50 for BRD3-2

Reference Compound IC50 for BRD3-2