BRPF3 Bromodomain Assay Service (AlphaScreen)

BRPF3-His Reader Domain Assay for compound screening and profiling using the AlphaScreen assay format to measure compound binding to the target.

Target Overview
CAT#

BRPF3

Enzyme

Human BRPF3

Synonyms

Bromodomain and PHD finger-containing protein 3, KIAA1286

Substrates

Histone H4 peptide (1-21) K5/8/12/16Ac

Assay Properties
Reaction

AlphaScreen Binding assay

Readout

Fluorescence

Reference Compound IC50s
Compounds IC50 (nM)
JQ-1 84,000
PFI-1 53,000
Bromosporine 13,000
Scientific Information

Q9ULD4 (http://www.uniprot.org/uniprot/Q9ULD4)

Screening Location

Malvern, USA

Further information

More information can be found on our website Reader Domain Assay Services.

Reference Compound IC50 for BRPF3

Reference Compound IC50 for BRPF3