CDC7/DBF4 Kinase Activity Assay Service

Activity-based CDC7/DBF4 kinase assay for compound screening and profiling via 33PanQinaseTM – assay technology

Target Overview
RBE Target ID

CDC7/DBF4

Enzyme

Human CDC7/DBF4, wt

HGNC

CDC7-DBF4

Manning ID

CDC7

Synonym

CDC7L1, HsCDC7, Hsk1, huCDC7, CDC7, HsCdc7, huCdc7, CDC7/DBF4

UniProt

O00311 (CDC7_HUMAN)

Kinase Type

Protein kinase

Kinase Group

Other

Assay Properties
Assay Format

33PanQinaseTM

Substrates

Histon H1, ATP

Reaction

Histon H1 + 33P-ATP = 33P-Histon H1 + ADP

Readout

Enzymatic activity

Technical Reference Compound IC50 value(s)
Compounds IC50 (nM)
Staurosporine 170
Sorafenib 10000
Sunitinib 100000
Screening Location

Freiburg, Germany

Further Information

More information can be found on our website Kinase Assays

Service and Product Availability
Screening Opportunities
FreeChoice CDC7/DBF4
355 wt Profiler Yes
355 IC50 wt Profiler Yes
Mutant Profiler Addon No
Lipid Kinase Profiler Addon No
IC50 Profiler No
Recombinant Protein Availability
Active recombinant protein Yes; ProQinaseTM – CDC7/DBF4
(Activity verified by 33PanQinaseTM-Assay)
Product Number 1513-1516-1
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