CSF1R Kinase Activity Assay Service

Activity-based CSF1R kinase assay for compound screening and profiling via 33PanQinaseTM – assay technology

Target Overview

RBE Target ID

CSF1R

Enzyme

Human CSF1R, wt

HGNC

CSF1R

Manning ID

FMS

Synonym

CSF1-R, C-FMS, CD115, CSFR, FIM2, CSF1R, CSF-1-R, FMS

UniProt

P07333 (CSF1R_HUMAN)

Kinase Type

Protein kinase

Kinase Group

TK

Assay Properties

Assay Format

33PanQinaseTM

Substrates

PolyEY, ATP

Reaction

PolyEY + 33P-ATP = 33P-PolyEY + ADP

Readout

Enzymatic activity

Technical Reference Compound IC50 value(s)
Compounds IC50 (nM)
Staurosporine 6
Sorafenib 2400
Sunitinb 760

Screening Location

Freiburg, Germany

Further Information

More information can be found on our website Kinase Assays

Service and Product Availability

Screening Opportunities
FreeChoice CSF1R
345 wt Profiler Yes
345 IC50 wt Profiler Yes
Mutant Profiler Addon No
Lipid Kinase Profiler Addon No
IC50 Profiler No
Recombinant Protein Availability
Active recombinant protein Yes; ProQinaseTM – CSF1R
(Activity verified by 33PanQinaseTM-Assay)
Product Number 0512-0000-1
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