NQO2 Assay Service

NQO2 (Ribosyldihydronicotinamide dehydrogenase [quinone]) assay for compound screening and profiling via fluorescence-based quantification of enzyme activity.

Target Overview
CAT#

NQO2

Enzyme

Human NQO2

Synonyms

NMOR2, NRH dehydrogenase [quinone] 2

Scientific Information
Assay Properties
Substrate

Menadione, dihydrobenzylnicotinamide (BNAH)

Reaction

1-Benzyl-1,4-dihydronicotinamide + menadione = 1-Benzyl-nicotinamide + menadiol

BNAH fluorescence, kinetic measurement

Readout

Enzymatic activity

Reference Compound IC50s
Compounds IC50 (nM)
Imatinib mesylate 183
Screening Location

Malvern, PA, USA

Further Information

More information can be found on our website NAD(P)H Dehydrogenase Assays (NQO)

Reference compound inhibition of NQO2

Reference compound inhibition of NQO2