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  1. Home
  2. List of Kinase Targets at US Facility

List of Biochemical Kinase Assays at US Facility

Target HGNC Reference Additional Synonyms Assay Format Protein_Lipid Bi-weekly Data
ABL1 ABL1 ABL, JTK7, p150, c-ABL, v-abl HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
ABL1 (E255K) ABL1 (E255K) ABL, JTK7, p150, c-ABL, v-abl HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ABL1 (E255V) ABL1 (E255V) ABL, JTK7, p150, c-ABL, v-abl HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ABL1 (F317I) ABL1 (F317I) ABL, JTK7, p150, c-ABL, v-abl HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ABL1 (F317L) ABL1 (F317L) ABL, JTK7, p150, c-ABL, v-abl HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ABL1 (G250E) ABL1 (G250E) ABL, JTK7, p150, c-ABL, v-abl HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ABL1 (H396P) ABL1 (H396P) ABL, JTK7, p150, c-ABL, v-abl HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ABL1 (M351T) ABL1 (M351T) ABL, JTK7, p150, c-ABL, v-abl HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ABL1 (Q252H) ABL1 (Q252H) ABL, JTK7, p150, c-ABL, v-abl HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ABL1 (T315I) ABL1 (T315I) ABL, JTK7, p150, c-ABL, v-abl HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ABL1 (V299L) ABL1 (V299L) ABL, JTK7, p150, c-ABL, v-abl HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ABL1 (Y253F) ABL1 (Y253F) ABL, JTK7, p150, c-ABL, v-abl HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ABL1 (Y253H) ABL1 (Y253H) ABL, JTK7, p150, c-ABL, v-abl HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ABL2/ARG ABL2 ABLL, ARG HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
ACK1 TNK2 ACK, p21cdc42Hs, Activated CDC42 kinase 1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
AKT1 AKT1 PKB, RAC, PRKBA, RAc-ALPHA HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
AKT1 (E17K) AKT1 (E17K) PKB, RAC, PRKBA, RAc-ALPHA HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
AKT2 AKT2 PRKBB, PKBBETA, RAc-BETA HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
AKT2 (E17K) AKT2 (E17K) PRKBB, PKBBETA, RAc-BETA HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
AKT3 AKT3 PKBG, PKB gamma, PRKBG, RAC-gamma, RAC-PK-gamma, STK-2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
AKT3 (E17K) AKT3 (E17K) PKBG, PKB gamma, PRKBG, RAC-gamma, RAC-PK-gamma, STK-2 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
AKT3 (G171R) AKT3 (G171R) PKBG, PKB gamma, PRKBG, RAC-gamma, RAC-PK-gamma, STK-2 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ALK ALK CD246, NBLST3 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
ALK (C1156Y) ALK (C1156Y) CD246, NBLST3 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ALK (F1174L) ALK (F1174L) CD246, NBLST3 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ALK (F1174L)-EML4 ALK (F1174L)-EML4 CD246, NBLST3, EML4-ALK (F1174L) HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ALK (F1174L)-NPM1 ALK (F1174L)-NPM1 CD246, NBLST3, NPM1-ALK (F1174L) HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ALK (F1174S) ALK (F1174S) CD246, NBLST3 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ALK (G1202R) ALK (G1202R) CD246, NBLST3 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ALK (G1269A) ALK (G1269A) CD246, NBLST3 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ALK (G1269S) ALK (G1269S) CD246, NBLST3 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ALK (L1152R) ALK (L1152R) CD246, NBLST3 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ALK (L1196M) ALK (L1196M) CD246, NBLST3 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ALK (R1275Q) ALK (R1275Q) CD246, NBLST3 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ALK (S1206R) ALK (S1206R) CD246, NBLST3 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ALK (T1151-L1152insT) ALK (T1151-L1152insT) CD246, NBLST3 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ALK (T1151M) ALK (T1151M) CD246, NBLST3 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ALK-KIF5B (Kex24Aex20) ALK-KIF5B CD246, NBLST3, KIF5B-ALK HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ALK-KLC1 (Kex8Aex20) ALK-KLC1 CD246, NBLST3, KCL1-ALK HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ALK-NPM1 ALK-NPM1 CD246, NBLST3, NPM1-ALK HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ALK-TFG ALK-TFG CD246, NBLST3, TFG-ALK HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ALK-TFG (Tex4Aex20) ALK-TFG CD246, NBLST3, TFG-ALK HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ALK-TPM1 ALK-TPM1 CD246, NBLST3, TPM1-ALK HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ALK-TPM3 ALK-TPM3 CD246, NBLST3, TPM3-ALK HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ALK1/ACVRL1 ACVRL1 ACVRLK1, ALK-1, ALK1, HHT, HHT2, ORW2, SKR3 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
ALK2 (Q207D) ACVR1 (Q207D) ACTRI, ACVRLK2, ALK2, SKR1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ALK2 (R206H) ACVR1 (R206H) ACTRI, ACVRLK2, ALK2, SKR1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ALK2/ACVR1 ACVR1 ACTRI, ACVRLK2, ALK2, SKR1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
ALK3/BMPR1A BMPR1A SKR5, CD292, ALK3, ACVRLK3 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
ALK4/ACVR1B ACVR1B ACTRIB, ACVRLK4, ALK4, SKR2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
ALK5/TGFBR1 TGFBR1 ALK5, ACVRLK4 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
ALK6/BMPR1B BMPR1B ALK6, CDw293 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
AMPK (A1/B1/G1) PRKAA1-PRKAB1-PRKAG1 AMPK (A1/B1/G1) HotSpot™ Protein kinase Bi-weekly Atypical Panel Data sheet
AMPK (A1/B1/G2) PRKAA1-PRKAB1-PRKAG2 AMPK (A1/B1/G2) HotSpot™ Protein kinase Bi-weekly Atypical Panel Data sheet
AMPK (A1/B1/G3) PRKAA1-PRKAB1-PRKAG3 AMPK (A1/B1/G3) HotSpot™ Protein kinase Bi-weekly Atypical Panel Data sheet
AMPK (A1/B2/G1) PRKAA1-PRKAB2-PRKAG1 AMPK (A1/B2/G1) HotSpot™ Protein kinase Bi-weekly Atypical Panel Data sheet
AMPK (A1/B2/G2) PRKAA1-PRKAB2-PRKAG2 AMPK (A1/B2/G2) HotSpot™ Protein kinase Bi-weekly Atypical Panel Data sheet
AMPK (A1/B2/G3) PRKAA1-PRKAB2-PRKAG3 AMPK (A1/B2/G3) HotSpot™ Protein kinase Bi-weekly Atypical Panel Data sheet
AMPK (A2/B1/G1) PRKAA2-PRKAB1-PRKAG1 AMPK (A2/B1/G1) HotSpot™ Protein kinase Bi-weekly Atypical Panel Data sheet
AMPK (A2/B1/G2) PRKAA2-PRKAB1-PRKAG2 AMPK (A2/B1/G2) HotSpot™ Protein kinase Bi-weekly Atypical Panel Data sheet
AMPK (A2/B1/G3) PRKAA2-PRKAB1-PRKAG3 AMPK (A2/B1/G3) HotSpot™ Protein kinase Bi-weekly Atypical Panel Data sheet
AMPK (A2/B2/G1) PRKAA2-PRKAB2-PRKAG1 AMPK (A2/B2/G1) HotSpot™ Protein kinase Bi-weekly Atypical Panel Data sheet
AMPK (A2/B2/G2) PRKAA2-PRKAB2-PRKAG2 AMPK (A2/B2/G2) HotSpot™ Protein kinase Bi-weekly Atypical Panel Data sheet
AMPK (A2/B2/G3) PRKAA2-PRKAB2-PRKAG3 AMPK (A2/B2/G3) HotSpot™ Protein kinase Bi-weekly Atypical Panel Data sheet
ARAF ARAF (Y301D/Y302D) A-RA, ARAF1, PKS2, RAFA1, ARAF YDYD HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
ARK5/NUAK1 NUAK1 KIAA0537, ARK5 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
ASK1/MAP3K5 MAP3K5 ASK1, MAPKKK5, MEKK5 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
ATM ATM TEL1, TELO1 HTRF Protein kinase Not included in any panel Data sheet
Aurora A AURKA AurA, AIK, ARK1, AURA, BTAK, STK15, AuroraA, Aurora A HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
Aurora B AURKB AurB, AIK2, AIM1, ARK2, AurB, IPL1, STK5, AuroraB, Aurora B HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
Aurora B (G160L) AURKB (G160L) AurB, AIK2, AIM1, ARK2, AurB, IPL1, STK5, AuroraB, Aurora B HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
Aurora C AURKC AurC, AIE2, AIK3, STK13, Aurora C, AuroraC HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
AXL AXL EC, UFO HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
AXL (R499C) AXL (R199C) EC, UFO HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
BLK BLK BLK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
BMPR2 BMPR2 BMPR-II, BMPR3, BMR2, BRK-3, PPH1, T-ALK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
BMX/ETK BMX ETK, PSCTK2, PSCTK3 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
BRAF BRAF B-Raf, B-raf-1, BRAF1, RAFB1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
BRAF (d485-489/P490Y) BRAF (d485-489/P490Y) B-Raf, B-raf-1, BRAF1, RAFB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
BRAF (G464V) BRAF (G464V) B-Raf, B-raf-1, BRAF1, RAFB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
BRAF (G469A) BRAF (G469A) B-Raf, B-raf-1, BRAF1, RAFB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
BRAF (K601E) BRAF (K601E) B-Raf, B-raf-1, BRAF1, RAFB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
BRAF (L597V) BRAF (L597V) B-Raf, B-raf-1, BRAF1, RAFB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
BRAF (R506_K507insVLR) BRAF (R506_K507insVLR) B-Raf, B-raf-1, BRAF1, RAFB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
BRAF (T599_V600insT) BRAF (T599_V600insT) B-Raf, B-raf-1, BRAF1, RAFB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
BRAF (V599E) BRAF (V600E) B-Raf, B-raf-1, BRAF1, RAFB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
BRAF (V600A) BRAF (V600A) B-Raf, B-raf-1, BRAF1, RAFB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
BRAF (V600D) BRAF (V600D) B-Raf, B-raf-1, BRAF1, RAFB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
BRAF (V600K) BRAF (V600K) B-Raf, B-raf-1, BRAF1, RAFB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
BRAF-FAM131B BRAF-FAM131B B-Raf, B-raf-1, BRAF1, RAFB1, FAM131B-BRAF HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
BRAF-KIAA1549 (Kex15Bex9) BRAF-KIAA1549 (Kex15Bex9) B-Raf, B-raf-1, BRAF1, RAFB1, KIAA1549-BRAF HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
BRAF-KIAA1549 (Kex16Bex9) BRAF-KIAA1549 (Kex16Bex9) B-Raf, B-raf-1, BRAF1, RAFB1, KIAA1549-BRAF HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
BRAF-SRGAP3 (Sex12Bex9) BRAF-SRGAP3 B-Raf, B-raf-1, BRAF1, RAFB1, SRGAP3-BRAF HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
BRK PTK6 BRK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
BRSK1 BRSK1 KIAA1811 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
BRSK2 BRSK2 C11orf7, FLJ41362, HUSSY-12, PEN11B, SAD1, STK29 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
BTK BTK AGMX1, AT, ATK, BPK, PSCTK1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
BTK (C481S) BTK (C481S) AGMX1, AT, ATK, BPK, PSCTK1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
BTK (E41K) BTK (E41K) AGMX1, AT, ATK, BPK, PSCTK1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
BTK (P190K) BTK (P190K) AGMX1, AT, ATK, BPK, PSCTK1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
BTK (T474I) BTK (T474I) AGMX1, AT, ATK, BPK, PSCTK1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
BTK (Y485F) BTK (Y485F) AGMX1, AT, ATK, BPK, PSCTK1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-KIT KIT C-Kit, PBT, CD117, SCFR, HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
c-KIT (A829P) KIT (A829P) C-Kit, PBT, CD117, SCFR, HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-KIT (d557-558) KIT (d557-558) C-Kit, PBT, CD117, SCFR, HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-KIT (D816E) KIT (D816E) C-Kit, PBT, CD117, SCFR, HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-KIT (D816F) KIT (D816F) C-Kit, PBT, CD117, SCFR, HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-KIT (D816H) KIT (D816H) C-Kit, PBT, CD117, SCFR, HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-KIT (D816I) KIT (D816I) C-Kit, PBT, CD117, SCFR, HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-KIT (D816V) KIT (D816V) C-Kit, PBT, CD117, SCFR, HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-KIT (D816Y) KIT (D816Y) C-Kit, PBT, CD117, SCFR, HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-KIT (D820E) KIT (D820E) C-Kit, PBT, CD117, SCFR, HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-KIT (D820Y) KIT (D820Y) C-Kit, PBT, CD117, SCFR, HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-KIT (K642E) KIT (K642E) C-Kit, PBT, CD117, SCFR, HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-KIT (T670I) KIT (T670I) C-Kit, PBT, CD117, SCFR, HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-KIT (V559A) KIT (V559A) C-Kit, PBT, CD117, SCFR, HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-KIT (V559D) KIT (V559D) C-Kit, PBT, CD117, SCFR, HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-KIT (V559D/T670I) KIT (V559D/T670I) C-Kit, PBT, CD117, SCFR, HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-KIT (V559D/V654A) KIT (V559D/V654A) C-Kit, PBT, CD117, SCFR, HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-KIT (V560G) KIT (V560G) C-Kit, PBT, CD117, SCFR, HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-KIT (V560G/D816V) KIT (V560G/D816V) C-Kit, PBT, CD117, SCFR, HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-KIT (V560G/N822K) KIT (V560G/N822K) C-Kit, PBT, CD117, SCFR, HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-KIT (V654A) KIT (V654A) C-Kit, PBT, CD117, SCFR, HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-KIT (Y823D) KIT (Y823D) C-Kit, PBT, CD117, SCFR, HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-MER MERTK MER, MER-PEN, RP38, c-MER HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
c-MER (A708S) MERTK (A708S) MER, MER-PEN, RP38, c-MER HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-MET MET c-MET, HGFR, RCCP2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
c-MET (D1228A) MET (D1228A) c-MET, HGFR, RCCP2 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-MET (D1228G) MET (D1228G) c-MET, HGFR, RCCP2 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-MET (D1228H) MET (D1228H) c-MET, HGFR, RCCP2 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-MET (D1228N) MET (D1228N) c-MET, HGFR, RCCP2 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-MET (D1228V) MET (D1228V) c-MET, HGFR, RCCP2 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-MET (D1228Y) MET (D1228Y) c-MET, HGFR, RCCP2 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-MET (F1200I) MET (F1200I) c-MET, HGFR, RCCP2 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-MET (G1163R) MET (G1163R) c-MET, HGFR, RCCP2 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-MET (H1094L) MET (H1094L) c-MET, HGFR, RCCP2 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-MET (H1094Y) MET (H1094Y) c-MET, HGFR, RCCP2 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-MET (K1244R) MET (K1244R) c-MET, HGFR, RCCP2 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-MET (L1195F) MET (L1195F) c-MET, HGFR, RCCP2 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-MET (L1195V) MET (L1195V) c-MET, HGFR, RCCP2 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-MET (M1250I) MET (M1250I) c-MET, HGFR, RCCP2 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-MET (M1250T) MET (M1250T) c-MET, HGFR, RCCP2 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-MET (P991S) MET (P991S) c-MET, HGFR, RCCP2 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-MET (T1173I) MET (T1173I) c-MET, HGFR, RCCP2 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-MET (T992I) MET (T992I) c-MET, HGFR, RCCP2 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-MET (V1092I) MET (V1092I) c-MET, HGFR, RCCP2 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-MET (Y1230A) MET (Y1230A) c-MET, HGFR, RCCP2 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-MET (Y1230C) MET (Y1230C) c-MET, HGFR, RCCP2 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-MET (Y1230D) MET (Y1230D) c-MET, HGFR, RCCP2 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-MET (Y1230H) MET (Y1230H) c-MET, HGFR, RCCP2 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-MET (Y1230S) MET (Y1230S) c-MET, HGFR, RCCP2 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-MET (Y1235D) MET (Y1235D) c-MET, HGFR, RCCP2 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-MET-KIF5B (Kex24Mex14) MET-KIF5B c-MET, HGFR, RCCP2, KIF5B-MET HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-MET-TFG (Tex5Mex15) MET-TFG c-MET, HGFR, RCCP2, TGF-MET HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-Src SRC ASV, SRC1, c-SRC, p60-Src HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
c-Src (T341M) SRC (T341M) ASV, SRC1, c-SRC, p60-Src HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
c-SRC (Y530F) SRC (Y530F) ASV, SRC1, c-SRC, p60-Src HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
CAMK1a CAMK1 CAMK1-PEN, CAMKI HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CAMK1b PNCK CAMK1b, MGC45419 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CAMK1d CAMK1D CKLiK, CaM-K1, CaMKID HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CAMK1g CAMK1G CLICKIII, VWS1, dJ272L16.1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CAMK2a CAMK2A CAMKA, KIAA0968 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CAMK2b CAMK2B CAM2, CAMK2, CAMKB, MGC29528 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CAMK2d CAMK2D CAMKD, MGC44911, CaMKII delta HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CAMK2g CAMK2G CAMK, CAMK-II, CAMKG, MGC26678 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CAMK4 CAMK4 CaMK-GR, MGC36771 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CAMKK1 CAMKK1 CAMKKA, DKFZp761M0423, MGC34095 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CAMKK2 CAMKK2 CAMKK, CAMKKB, KIAA0787, MGC15254 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CDC7/DBF4 CDC7-DBF4 CDC7L1, HsCdc7, HsCDC7, Hsk1, huCdc7 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CDK1/cyclin A CDK1-CCNA2 CDC2, p34 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CDK1/cyclin B CDK1-CCNB1 CDC2, p34 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CDK1/cyclin E CDK1-CCNE1 CDC2, p34 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CDK12 (R722C)/cyclin K* CDK12 (R722C)-CCNK CRKRS, CRK7 HotSpot™ Protein kinase Not included in any panel Data sheet
CDK12/cyclin K* CDK12-CCNK CRKRS, CRK7 HotSpot™ Protein kinase Not included in any panel Data sheet
CDK13/cyclin K* CDK13-CCNK CDC2L, CDC2L5, CHED HotSpot™ Protein kinase Not included in any panel Data sheet
CDK14/cyclin Y (PFTK1) CDK14-CCNY PFTAIRE1, PFTK1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CDK16/cyclin Y CDK16-CCNY PCTAIRE1, PCTAIRE, PCTGAIRE, PCTK1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CDK17/cyclin Y CDK17-CCNY PCTAIRE2, PCTK2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CDK18/cyclin Y CDK18-CCNY PCTAIRE, PCTAIRE3, PCTK3 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CDK19/cyclin C* CDK19-CCNC CDC2L6, CDK11 HotSpot™ Protein kinase Not included in any panel Data sheet
CDK2/cyclin A CDK2-CCNA2 p33 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CDK2/cyclin A1 CDK2-CCNA1 p33 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CDK2/cyclin E CDK2-CCNE1 p33 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CDK2/cyclin E2 CDK2-CCNE2 p33 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CDK2/cyclin O CDK2-CCNO p33 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CDK3/cyclin E CDK3-CCNE1 CDKN3 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CDK3/cyclin E2 CDK3-CCNE2 CDKN3 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CDK4/cyclin D1 CDK4-CCND1 CMM3, PSK-J3 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CDK4/cyclin D2 CDK4-CCND2 CMM3, PSK-J3 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CDK4/cyclin D3 CDK4-CCND3 CMM3, PSK-J3 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CDK5/p25 CDK5-CDK5R1 (p25) PSSALRE HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CDK5/p35 CDK5-CDK5R1 PSSALRE HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CDK6/cyclin D1 CDK6-CCND1 PLSTIRE HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CDK6/cyclin D2 CDK6-CCND2 PLSTIRE HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CDK6/cyclin D3 CDK6-CCND3 PLSTIRE HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CDK7/cyclin H CDK7-CCNH-MNAT1 CAK1, CDKN7, STK1, p39MO15 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CDK8/cyclin C CDK8-CCNC K35 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CDK9/cyclin K CDK9-CCNK C-2k, CDC2L4, PITALRE, TAK, CDC2-related kinase HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CDK9/cyclin T1 CDK9-CCNT1 C-2k, CDC2L4, PITALRE, TAK, CDC2-related kinase HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CDK9/cyclin T2 CDK9-CCNT2 C-2k, CDC2L4, PITALRE, TAK, CDC2-related kinase HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CHK1 CHEK1 CHEK1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CHK2 CHEK2 CDS1, HuCds1, PP1425, RAD53, bA444G7 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CHK2(I157T) CHEK2 (I157T) CDS1, HuCds1, PP1425, RAD53, bA444G7 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
CK1a1 CSNK1A1 CK1, HLCDGP1, PRO2975, CK1-alpha1, CK1alpha1, CK1a1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CK1a1L CSNK1A1L CK1-alpha1 like HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CK1d CSNK1D HCKID, CK1-delta, CK1d, CK1delta HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CK1epsilon CSNK1E CKIe, HCKIE, MGC10398, CK1-epsilon HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CK1epsilon (R178C) CSNK1E (R178C) CKIe, HCKIE, MGC10398, CK1-epsilon HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
CK1g1 CSNK1G1 CK1-gamma1, CK1gamma1, CK1g1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CK1g2 CSNK1G2 CK1g2, CK1-gamma2, CK1gamma2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CK1g3 CSNK1G3 CK1-gamma3, CK1gamma3 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CK2a CSNK2A1 CKII, CK2A1, CK2-alpha1, CK2alpha1, CK2a HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CK2a2 CSNK2A2 CK2-alpha2, CK2alpha2, CK2a2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CLK1 CLK1 CLK, CLK/STY HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CLK2 CLK2 MGC61500, hCLK2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CLK3 CLK3 PHCLK3, PHCLK3/152, CDc-like kinase 3 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CLK4 CLK4 DKFZp686A20267, CDc-like kinase 4 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
COT1/MAP3K8 MAP3K8 COT1, EST, ESTF, TPL2, Tpl-2, COT HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CSK CSK CSK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
CTK/MATK MATK CHK, CTK, DKFZp434N1212, HHYLTK, HYL, Lsk, MGC1708, MGC2101 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
DAPK1 DAPK1 DAPK1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
DAPK2 DAPK2 DRP-1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
DCAMKL1 DCLK1 DCLK, KIAA0369 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
DCAMKL2 DCLK2 DCDC3, DCK2, MGC45428, KIAA0369 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
DDR1 DDR1 CAK, CD167, DDR, EDDR1, MCK10, NEP HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
DDR2 DDR2 MIG20a, NTRKR3, TKT, TYRO10 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
DDR2 (N456S) DDR2 (N456S) MIG20a, NTRKR3, TKT, TYRO10 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
DDR2 (T654M) DDR2 (T654M) MIG20a, NTRKR3, TKT, TYRO10 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
DGKA* DGKA DAGK1, DAGK, DGK-alpha ADP-Glo Lipid kinase Not included in any panel Please inquire
DGKB* DGKB DAGK2, KIAA0718, DGK-beta ADP-Glo Lipid kinase Not included in any panel Please inquire
DGKD* DGKD DGK-delta, KIAA0145 ADP-Glo Lipid kinase Not included in any panel Please inquire
DGKE* DGKE DAGK5, DGK-epsilon ADP-Glo Lipid kinase Not included in any panel Please inquire
DGKG* DGKG DAGK3, DGK-gamma ADP-Glo Lipid kinase Not included in any panel Please inquire
DGKH* DGKH DGK-eta ADP-Glo Lipid kinase Not included in any panel Please inquire
DGKI* DGKI DGK-iota ADP-Glo Lipid kinase Not included in any panel Please inquire
DGKK* DGKK DGK-kappa ADP-Glo Lipid kinase Not included in any panel Please inquire
DGKQ* DGKQ DAGK4, DGK-theta ADP-Glo Lipid kinase Not included in any panel Please inquire
DGKZ* DGKZ DAGK6, DGK-zeta ADP-Glo Lipid kinase Not included in any panel Please inquire
DLK/MAP3K12 MAP3K12 DLK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
DMPK DMPK DMPK1, DM, DM1, DM1PK, DMK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
DMPK2/CDC42BPG CDC42BPG DMPK2, HSMDPKIN, KAPPA-200, HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
DNA-PK PRKDC DNPK1, HYRC, p350, DNAPK, DNA-PK HotSpot™ Protein kinase Bi-weekly Atypical Panel Data sheet
DRAK1/STK17A STK17A DRAK1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
DYRK1/DYRK1A DYRK1A DYRK, DYRK1, HP86, MNB, MNBH HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
DYRK1B DYRK1B MIRK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
DYRK2 DYRK2 DYRK2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
DYRK3 DYRK3 DYRK5, RED, REDK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
DYRK4 DYRK4 DYRK4 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
EEF2K EEF2K HSU93850, MGC45041, eEF-2K HotSpot™ Protein kinase Bi-weekly Atypical Panel Data sheet
EGFR EGFR ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
EGFR (A763_Y764insFHEA) EGFR (A763_Y764insFHEA) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (A763_Y764insFQEA) EGFR (A763_Y764insFQEA) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (A767_S768insTLA) EGFR (A767_S768insTLA) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (C775S/T790M/L858R) EGFR (C775S/T790M/L858R) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (C797A) EGFR (C797A) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (C797G/L858R) EGFR (C797G/L858R) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (C797S) EGFR (C797S) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (C797S/L858R) EGFR (C797S/L858R) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (d746) EGFR (d746) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (d746-750) EGFR (d746-750) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (d746-750/C775S /T790M /L858R) EGFR (d746-750/C775S/T790M/L858R) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (d746-750/C797A) EGFR (d746-750/C797A) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (d746-750/C797S) EGFR (d746-750/C797S) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (d746-750/G724S) EGFR (d746-750/G724S) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (d746-750/S768I) EGFR (d746-750/S768I) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (d746-750/T790M) EGFR (d746-750/T790M) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (d746-750/T790M/C797S) EGFR (d746-750/T790M/C797S) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (d746-750/T790M/C797S/L858R) EGFR (d746-750/T790M/C797S/L858R) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (d747-749) EGFR (d747-749) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (d747-749/A750P) EGFR (d747-749/A750P) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (d747-752/P753S) EGFR (d747-752/P753S) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (d752-759) EGFR (d752-759) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (D761Y) EGFR (D761Y) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (D770_N771insNPG) EGFR (D770_N771insNPG) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (D770_N771insNPG/T790M) EGFR (D770_N771insNPG/T790M) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (D770GY) EGFR (D770GY) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (G719C) EGFR (G719C) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (G719D) EGFR (G719D) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (G719S) EGFR (G719S) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (K716A) EGFR (K716A) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (K716A/C797S/L858R) EGFR (K716A/C797S/L858R) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (K716A/T790M/C797S/L858R) EGFR (K716A/T790M/C797S/L858R) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (K716Q/L718Q) EGFR (K716Q/L718Q) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (K728A) EGFR (K728A) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (K728A/T790M/C797S/L858R) EGFR (K728A/T790M/C797S/L858R) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (L718Q) EGFR (L718Q) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (L747S) EGFR (L747S) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (L792F) EGFR (L792F) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (L792F/L858R) EGFR (L792F/L858R) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (L792H) EGFR (L792H) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (L792H/C797S/L858R) EGFR (L792H/C797S/L858R) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (L792H/L858R) EGFR (L792H/L858R) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (L858R) EGFR (L858R) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (L858R/T790M) EGFR (T790M/L858R) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (L861Q) EGFR (L861Q) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (N771_P772insH) EGFR (N771_P772insH) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (R999A) EGFR (R999A) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (T790M) EGFR (T790M) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (T790M/C797S /L858R) EGFR (T790M/C797S/L858R) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (T790M/C797S) EGFR (T790M/C797S) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (T790M/L792F/C797S/L858R) EGFR (T790M/L792F/C797S/L858R) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (T790M/L792F/L858R) EGFR (T790M/L792F/L858R) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (T790M/L792H/C797S/L858R) EGFR (T790M/L792H/C797S/L858R) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (T790M/L792H/L858R) EGFR (T790M/L792H/L858R) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EGFR (V769_D770insGE) EGFR (V769_D770insGE) EGF-R, ERBB, mENA, ERBB1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
EIF2AK1 EIF2AK1 HCR, HRI, EIF2AK1 HotSpot™ Protein kinase Bi-weekly Atypical Panel Data sheet
EIF2AK2 EIF2AK2 PKR, PRKR HotSpot™ Protein kinase Bi-weekly Atypical Panel Data sheet
EIF2AK3 EIF2AK3 DKFZp781H1925, PEK, PERK, WRS HotSpot™ Protein kinase Bi-weekly Atypical Panel Data sheet
EIF2AK4/GCN2 EIF2AK4 GCN2 HotSpot™ Protein kinase Bi-weekly Atypical Panel Data sheet
EPHA1 EPHA1 EPH, EPHT, EPHT1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
EPHA2 EPHA2 ECK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
EPHA3 EPHA3 ETK, ETK1, HEKECK, HEK4, TYRO4 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
EPHA4 EPHA4 HEK8, SEK, TYRO1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
EPHA5 EPHA5 CEK7, EHK1,HEK7, HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
EPHA6 EPHA6 EHK2, EHK-2, EPA6 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
EPHA7 EPHA7 EHK3, HEK11 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
EPHA8 EPHA8 EEK, HEK3, KIAA1459 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
EPHB1 EPHB1 ELK, NET, Hek6, EPHT2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
EPHB2 EPHB2 DRT, ERK, Hek5, EPHT3, Tyro5 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
EPHB3 EPHB3 ETK2, HEK2, TYRO6 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
EPHB4 EPHB4 HTK, MYK1, TYRO11 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
ERBB2 (A775_G776insYVMA) ERBB2 (A775_G776insYVMA) NEU, NGL, HER2, TKR1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ERBB2 (D769H) ERBB2 (D769H) NEU, NGL, HER2, TKR1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ERBB2 (D769Y) ERBB2 (D769Y) NEU, NGL, HER2, TKR1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ERBB2 (P1170A) ERBB2 (P1170A) NEU, NGL, HER2, TKR1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ERBB2 (P780-Y781insGSP) ERBB2 (P780-Y781insGSP) NEU, NGL, HER2, TKR1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ERBB2 (R896C) ERBB2 (R896C) NEU, NGL, HER2, TKR1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ERBB2 (V777_G778insCG) ERBB2 (V777_G778insCG) NEU, NGL, HER2, TKR1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ERBB2 (V777L) ERBB2 (V777L) NEU, NGL, HER2, TKR1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ERBB2/HER2 ERBB2 NEU, NGL, HER2, TKR1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
ERBB4/HER4 ERBB4 HER4 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
ERK1/MAPK3 MAPK3 ERT2, HS44KDAP, HUMKER1A, P44ERK1, P44MAPK, PRKM3 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
ERK2/MAPK1 MAPK1 ERK2, ERT1, P42MAPK, PRKM1, HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
ERK5/MAPK7 CD* MAPK7 (CD) BMK1, ERK4, PRKM7 HotSpot™ Protein kinase Not included in any panel Data sheet
ERK5/MAPK7 FL MAPK7 BMK1, ERK4, PRKM7 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
ERK7/MAPK15 MAPK15 ERK8 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
ERN1 (R727A) ERN1 (R727A) IRE1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ERN1 (R728A) ERN1 (R728A) IRE1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ERN1/IRE1 ERN1 IRE1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
ERN2/IRE2 ERN2 IRE2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
FAK/PTK2 PTK2 FAK, FADK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
FER FER TYK3, c-FER, p94-FER HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
FES/FPS FES FPS HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
FGFR1 FGFR1 H2, H3, H4, H5, CEK, FLG, FLT2, KAL2, BFGFR, C-FGR, N-SAM HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
FGFR1(V561M) FGFR1 (V561M) H2, H3, H4, H5, CEK, FLG, FLT2, KAL2, BFGFR, C-FGR, N-SAM HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
FGFR1OP- FGFR1 CEP43-FGFR1 FOP, CEP43, FGFR1-FGFR1OP HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
FGFR2 FGFR2 BEK, BFR-1, CD332, CEK3, CFD1, ECT1, JWS, KGFR, KSAM, K-SAM, TK14, TK25 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
FGFR2 (C491A) FGFR2 (C491A) BEK, BFR-1, CD332, CEK3, CFD1, ECT1, JWS, KGFR, KSAM, K-SAM, TK14, TK25 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
FGFR2 (C491F) FGFR2 (C491F) BEK, BFR-1, CD332, CEK3, CFD1, ECT1, JWS, KGFR, KSAM, K-SAM, TK14, TK25 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
FGFR2 (C491S) FGFR2 (C491S) BEK, BFR-1, CD332, CEK3, CFD1, ECT1, JWS, KGFR, KSAM, K-SAM, TK14, TK25 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
FGFR2 (E565G) FGFR2 (E565G) BEK, BFR-1, CD332, CEK3, CFD1, ECT1, JWS, KGFR, KSAM, K-SAM, TK14, TK25 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
FGFR2 (K526E) FGFR2 (K526E) BEK, BFR-1, CD332, CEK3, CFD1, ECT1, JWS, KGFR, KSAM, K-SAM, TK14, TK25 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
FGFR2 (K641R) FGFR2 (K641R) BEK, BFR-1, CD332, CEK3, CFD1, ECT1, JWS, KGFR, KSAM, K-SAM, TK14, TK25 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
FGFR2 (K659N) FGFR2 (K659N) BEK, BFR-1, CD332, CEK3, CFD1, ECT1, JWS, KGFR, KSAM, K-SAM, TK14, TK25 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
FGFR2 (N549H) FGFR2 (N549H) BEK, BFR-1, CD332, CEK3, CFD1, ECT1, JWS, KGFR, KSAM, K-SAM, TK14, TK25 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
FGFR2 (R612T) FGFR2 (R612T) BEK, BFR-1, CD332, CEK3, CFD1, ECT1, JWS, KGFR, KSAM, K-SAM, TK14, TK25 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
FGFR2 (V564F) FGFR2 (V564F) BEK, BFR-1, CD332, CEK3, CFD1, ECT1, JWS, KGFR, KSAM, K-SAM, TK14, TK25 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
FGFR3 FGFR3 ACH, CD333, CEK2, HSFGFR3EX, JTK4 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
FGFR3 (G697C) FGFR3 (G697C) ACH, CD333, CEK2, HSFGFR3EX, JTK4 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
FGFR3 (K650E) FGFR3 (K650E) ACH, CD333, CEK2, HSFGFR3EX, JTK4 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
FGFR3 (K650M) FGFR3 (K650M) ACH, CD333, CEK2, HSFGFR3EX, JTK4 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
FGFR3 (K650Q) FGFR3 (K650Q) ACH, CD333, CEK2, HSFGFR3EX, JTK4 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
FGFR3 (V555M) FGFR3 (V555M) ACH, CD333, CEK2, HSFGFR3EX, JTK4 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
FGFR4 FGFR4 TKF, JTK2, MGC20292 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
FGFR4 (N535K) FGFR4 (N535K) TKF, JTK2, MGC20292 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
FGFR4 (V550E) FGFR4 (V550E) TKF, JTK2, MGC20292 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
FGFR4 (V550L) FGFR4 (V550L) TKF, JTK2, MGC20292 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
FGFR4 (V550M) FGFR4 (V550M) TKF, JTK2, MGC20292 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
FGR FGR SRC2, c-fgr, p55c-fgr HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
FLT1/VEGFR1 FLT1 FLT, VEGFR1, FLT1, VEGF-R1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
FLT3 FLT3 FLK2, STK1, CD135 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
FLT3 (D835Y) FLT3 (D835Y) FLK2, STK1, CD135 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
FLT3 (F594_R595insR) FLT3 (F594_R595insR) FLK2, STK1, CD135 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
FLT3 (F594_R595insREY) FLT3 (F594_R595insREY) FLK2, STK1, CD135 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
FLT3 (ITD) FLT3 (ITD) FLK2, STK1, CD135 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
FLT3 (ITD)-NPOS FLT3 (ITD)-NPOS FLK2, STK1, CD135 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
FLT3 (ITD)-W51 FLT3 (ITD)-W51 FLK2, STK1, CD135 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
FLT3 (R595_E596insEY) FLT3 (R595_E596insEY) FLK2, STK1, CD135 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
FLT3 (Y591_V592insVDFREYEYD) FLT3 (Y591_V592insVDFREYEYD) FLK2, STK1, CD135 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
FLT4/VEGFR3 FLT4 VEGFR3, PCL, VEGF-R3 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
FMS CSF1R C-FMS, CD115, CSF-1-R, CSFR, FIM2, FMS, CSF1R HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
FRK/PTK5 FRK PTK5, GTK, RAK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
FYN FYN SLK, SYN, p59-Fyn HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
FYN (Y531F) FYN (Y531F) SLK, SYN, p59-Fyn HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
GCK/MAP4K2 MAP4K2 BL44, GCK, RAB8IP HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
GLK/MAP4K3 MAP4K3 GLK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
GRK1 GRK1 RHOK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
GRK2 GRK2 ADRBK1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
GRK3 GRK3 ADRBK2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
GRK4 GRK4 GPRK2L, GPRK4, GRK4a, IT11 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
GRK5 GRK5 GPRK5 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
GRK6 GRK6 GPRK6, FLJ32135 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
GRK7 GRK7 GPRK7 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
GSK3a GSK3A GSK3alpha, GSK3a HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
GSK3b GSK3B GSK3beta, GSK3b HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
Haspin GSG2 GSG2, Haspin HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
HCK HCK JTK9 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
HGK/MAP4K4 MAP4K4 HGK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
HIPK1 HIPK1 KIAA0630, MGC26642, MGC33446, Myak, Nbak2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
HIPK2 HIPK2 PRO0593 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
HIPK3 HIPK3 ANPK, DYRK6, FIST, FIST3, PKY, YAK1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
HIPK4 HIPK4 FLJ32818 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
HPK1/MAP4K1 MAP4K1 HPK1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
IGF1R IGF1R JTK13, IGFR, CD221 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
IKKa/CHUK CHUK IKBKA, IKK1, IKKA, NFKBIKA, TCF16, IKK-alpha, IKKalpha, IKKa HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
IKKb/IKBKB IKBKB IKK2, IKKB, NFKBIKB, IKK-beta, IKKbeta HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
IKKe/IKBKE IKBKE IKKI, IKK-i, KIAA0151, IKK-epsilon, IKKepsilon HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
IR INSR IR HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
IRAK1 IRAK1 Pelle HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
IRAK2 IRAK2 Interleukin-1 receptor-associated kinase-like 2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
IRAK4 IRAK4 REN64 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
IRR/INSRR INSRR IRR HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
ITK ITK EMT 2, LYK 2, PSCTK2 2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
JAK1 JAK1 (aa866-1154) JAK1A, JAK1B, JTK3 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
JAK2 JAK2 JAK2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
JAK2 (V617F) JAK2 (V617F) JAK2 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
JAK2 JH1&2* JAK2 (JH1&2) JAK2 HotSpot™ Protein kinase Not included in any panel Data sheet
JAK3 JAK3 JAKL, L-JAK, LJAK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
JNK1 MAPK8 PRKM8, SAPK1, JNK1-alpha1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
JNK2 MAPK9 PRKM9, SAPK, p54a, JNK-alpha2, JNK2A, JNK2B HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
JNK3 MAPK10 JNK3A, PRKM10, p493F12 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
KDR/VEGFR2 KDR VEGFR2, FLK1, VEGF-R2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
KHS/MAP4K5 MAP4K5 KHS1, GCKR, KHS, MAPKKKK5 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
KSR1 KSR1 Kinase suppressor of Ras 1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
KSR1 (A635F) KSR1 (A635F) Kinase suppressor of Ras 1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
KSR1 (L639F) KSR1 (L639F) Kinase suppressor of Ras 1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
KSR2 KSR2 Kinase suppressor of Ras 2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
KSR2 (R676S) KSR2 (R676S) Kinase suppressor of Ras 2 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
LATS1 LATS1 WARTS, wts HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
LATS2 LATS2 FLJ13161, LATS HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
LCK LCK LCK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
LCK2/ICK CILK1 LCK2, ICK, MRK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
LIMK1 LIMK1 LIMK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
LIMK2 LIMK2 LIMK2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
LKB1 STK11 LKB1, PJS HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
LOK/STK10 STK10 LOK, PRO2729 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
LRRK2 LRRK2 PARK8, ROCO2, FLJ45829, DKFZp434H2111 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
LRRK2 (G2019S) LRRK2 (G2019S) PARK8, ROCO2, FLJ45829, DKFZp434H2111 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
LRRK2 (I2020T) LRRK2 (I2020T) PARK8, ROCO2, FLJ45829, DKFZp434H2111 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
LRRK2 (R1441C) LRRK2 (R1441C) PARK8, ROCO2, FLJ45829, DKFZp434H2111 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
LYN LYN JTK8 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
LYNB LYN (d23-43) JTK8 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MAK MAK MAK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MAPKAPK2 MAPKAPK2 MAPKAPK2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MAPKAPK3 MAPKAPK3 3PK, MAPKAP, MAPKAP3 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MAPKAPK5/PRAK MAPKAPK5 PRAK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MARK1 MARK1 KIAA1477 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MARK2/PAR-1Ba MARK2 EMK1, MGC99619, PAR-1Ba, ELKL HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MARK3 MARK3 CTAK1, KP78, PAR1A HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MARK4 MARK4 KIAA1860, MARKL1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MAST3 MAST3 Microtubule-associated serine/threonine-protein kinase 3, KIAA0561 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MASTL MASTL GLW, GREATWALL, GWL, hGWL, THC2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MEK1 MAP2K1 MAPKK1, MKK1, PRKMK1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MEK1 (P124L) MAP2K1 (P124L) MAPKK1, MKK1, PRKMK1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
MEK2 MAP2K2 MAPKK2, MKK2, PRKMK2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MEK3 MAP2K3 MEK3 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MEK5 MAP2K5 MAPKK5, MKK5, PRKMK5 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MEKK1 MAP3K1 MAPKKK1, MEKK, MEKK1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MEKK2 MAP3K2 MAPKKK2, MEKK2B HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MEKK3 MAP3K3 MAPKKK3, MEK kinase3 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MEKK6 MAP3K6 ASK2, MAPKKK6 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MELK MELK KIAA0175, PK38 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MELK (T460M) MELK (T460M) KIAA0175, PK38 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
MINK/MINK1 MINK1 B55, YSK2, MAP4K6, ZC3, MINK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MKK4 MAP2K4 JNKK, JNKK1, MAPKK4, MEK4, PRKMK4, SEK, SERK1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MKK6 MAP2K6 MAPKK6, MEK6, PRKMK6, SAPKK3 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MKK7 MAP2K7 MAPKK7, MEK7, PRKMK7 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MLCK/MYLK MYLK smMLCK, FLJ12216, KRP, MLCK, MLCK108, MLCK210 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MLCK2/MYLK2 MYLK2 KMLC, skMLCK, MLCK2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MLK1/MAP3K9 MAP3K9 MLK1, PRKE1, MEKK9 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MLK2/MAP3K10 MAP3K10 MLK2, MST, MEKK10 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MLK3/MAP3K11 MAP3K11 MGC17114, MLK-3, PTK1, SPRK, MLK3 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MLK4 MAP3K21 KIAA1804 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MNK1 MKNK1 MNK1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MNK2 MKNK2 MNK2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MRCKa/CDC42BPA CDC42BPA MRCK-alpha, MRCKa HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MRCKb/CDC42BPB CDC42BPB MRCK-beta, MRCKb HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MSK1/RPS6KA5 RPS6KA5 MSK1, RLPK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MSK2/RPS6KA4 RPS6KA4 MSK2, RSK-B HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MSSK1/STK23 SRPK3 MSSK1, MGC102944, STK23 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MST1/STK4 STK4 MST1, KRS2, YSK3 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MST2/STK3 STK3 MST2, KRS1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MST3/STK24 STK24 MST3 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MST4 STK26 MASK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
mTOR/FRAP1 MTOR FRAP1, FRAP, FRAP2, RAFT1, RAPT1 HotSpot™ Protein kinase Bi-weekly Atypical Panel Data sheet
MUSK MUSK MUSK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MYLK3 MYLK3 caMLCK, MLCK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MYLK4 MYLK4 Myosin light chain kinase family member 4 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MYO3A MYO3A Myosin-IIIa HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
MYO3b MYO3B MYO3b HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
NEK1 NEK1 KIAA1901, NY-REN-55, HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
NEK11 NEK11 FLJ23495 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
NEK2 NEK2 NLK1, HsPK21, HsPK 21 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
NEK3 NEK3 HSPK36, MGC29949 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
NEK4 NEK4 NRK2, STK2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
NEK5 NEK5 MGC75495 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
NEK6 NEK6 SID6-1512 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
NEK7 NEK7 NEK7 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
NEK8 NEK8 NEK8 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
NEK9 NEK9 DKFZp434D0935, MGC16714, NERCC, HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
NIK/MAP3K14* MAP3K14 NIK, FTDCR1B, HS, HSNIK HotSpot™ Protein kinase Not included in any panel Data sheet
NIM1 NIM1K NIM1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
NLK NLK NLK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
OSR1/OXSR1 OXSR1 OSR1, KIAA1101 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
p38a (T106M) MAPK14 (T106M) p38-alpha, CSBP, CSBP1, p38alpha, p38a HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
P38a/MAPK14 MAPK14 p38-alpha, CSBP, CSBP1, p38alpha, p38a HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
P38b/MAPK11 MAPK11 p38-beta, P38BETA2, PRKM11, SAPK2, p38beta, p38b HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
P38d/MAPK13 MAPK13 p38-delta, PRKM13, SAPK4, p38delta, p38d HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
P38g/MAPK12 MAPK12 p38-gamma, ERK3, ERK5, ERK6, p38gamma, p38g HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
P70S6K/RPS6KB1 RPS6KB1 S6K, STK14A, P70S6K HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
P70S6Kb/RPS6KB2 RPS6KB2 KLS, P70-beta-1, P70-beta-2, S6K-beta2, S6K2, SRK, p70S6Kb, S6K-beta, S6Kbeta HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PAK1 PAK1 PAKalpha HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PAK2 PAK2 PAK65, PAKgamma HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PAK2 (Y443N) PAK2 (Y443N) PAK-2, PAK65, Gamma-PAK, S6/H4 kinase HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
PAK3 PAK3 MRX30, OPHN3, PAK3beta, bPAK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PAK4 PAK4 PAK4 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PAK5 PAK5 PAK7, PAK5, KIAA1264, MGC26232 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PAK6 PAK6 PAK6, PAK5 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PASK PASK DKFZP434O051, DKFZp686P2031, KIAA0135, PASKIN, STK3 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PBK/TOPK PBK TOPK, SPK, Nori-3, FLJ14385 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PDGFRa PDGFRA PDGFRalpha, PDGFR2, CD140a HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PDGFRa(D842V) PDGFRA (D842V) PDGFRalpha, PDGFR2, CD140a HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
PDGFRa(G680R) PDGFRA (G680R) PDGFRalpha, PDGFR2, CD140a HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
PDGFRa(T674I) PDGFRA (T674I) PDGFRalpha, PDGFR2, CD140a HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
PDGFRa(V561D) PDGFRA (V561D) PDGFRalpha, PDGFR2, CD140a HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
PDGFRa-FIP1L1 PDGFRA-FIP1L1 PDGFRalpha, PDGFR2, CD140a, FIP1L1-PDGFRA HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
PDGFRb PDGFRB PDGFRbeta, JTK12, PDGFR, CD140B, PDGFR1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PDGFRb-TPM3 PDGFRB-TPM3 PDGFRbeta, JTK12, PDGFR, CD140B, PDGFR1, TPM3-PDGFRB HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
PDK1/PDHK1 PDK1 PDHK1, Pyruvate dehydrogenase kinase HotSpot™ Protein kinase Bi-weekly Atypical Panel Data sheet
PDK1/PDPK1 PDPK1 PDK1, PKB-like, 3-phosphoinositide-dependent protein kinase 1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PDK2/PDHK2 PDK2 PDHK2 HotSpot™ Protein kinase Bi-weekly Atypical Panel Data sheet
PDK3/PDHK3 PDK3 PDHK3 HotSpot™ Protein kinase Bi-weekly Atypical Panel Data sheet
PDK4/PDHK4 PDK4 PDHK4 HotSpot™ Protein kinase Bi-weekly Atypical Panel Data sheet
PEAK1 PEAK1 PEAK1, KIAA2002 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PHKg1 PHKG1 PHKg1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PHKg2 PHKG2 PHKg2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PI3K (p110a(E542K)/p85a) PIK3CA (E542K)-PIK3R1 MGC142161, MGC142163, p110-alpha, PI3K, PI3K-alpha ADP-Glo Lipid kinase Bi-weekly Lipid Kinase Panel Data sheet
PI3K (p110a(E545K)/p85a) PIK3CA (E545K)-PIK3R1 MGC142161, MGC142163, p110-alpha, PI3K, PI3K-alpha ADP-Glo Lipid kinase Bi-weekly Lipid Kinase Panel Data sheet
PI3K (p110a(H1047R)/p85a) PIK3CA (H1047R)-PIK3R1 MGC142161, MGC142163, p110-alpha, PI3K, PI3K-alpha ADP-Glo Lipid kinase Bi-weekly Lipid Kinase Panel Data sheet
PI3K (p110a/p65a) PIK3CA-PIK3R1/p65a MGC142161, MGC142163, p110-alpha, PI3K, PI3K-alpha ADP-Glo Lipid kinase Bi-weekly Lipid Kinase Panel Data sheet
PI3Ka (p110a/p85a) PIK3CA-PIK3R1 MGC142161, MGC142163, p110-alpha, PI3K, PI3K-alpha ADP-Glo Lipid kinase Bi-weekly Lipid Kinase Panel Data sheet
PI3Kb (p110b/p85a) PIK3CB-PIK3R1 PI3K, PI3KBETA, PIK3C1, p110-beta ADP-Glo Lipid kinase Bi-weekly Lipid Kinase Panel Data sheet
PI3KC2a PIK3C2A CPK, MGC142218, PI3-K-C2A ADP-Glo Lipid kinase Bi-weekly Lipid Kinase Panel Data sheet
PI3KC3 PIK3C3 MGC61518, PI3-kinase type 3, PI3K type 3, Vps34 ADP-Glo Lipid kinase Bi-weekly Lipid Kinase Panel Data sheet
PI3Kd (p110d/p85a) PIK3CD-PIK3R1 p110D, P110DELTA, PI3K, PI3K-delta, p110-delta ADP-Glo Lipid kinase Bi-weekly Lipid Kinase Panel Data sheet
PI3Kg (p110g) PIK3CG p120-PI3K, PI3CG, PI3K, PI3Kgamma, p110-gamma ADP-Glo Lipid kinase Bi-weekly Lipid Kinase Panel Data sheet
PI4K2A PI4K2A PI4KII, PIK42A, RP11-548K23.6 ADP-Glo Lipid kinase Bi-weekly Lipid Kinase Panel Data sheet
PI4Ka PI4KA PIK4CA ADP-Glo Lipid kinase Bi-weekly Lipid Kinase Panel Data sheet
PI4Kb PI4KB PIK4CB, NPIK ADP-Glo Lipid kinase Bi-weekly Lipid Kinase Panel Data sheet
PIM1 PIM1 PIM HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PIM2 PIM2 PIM2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PIM3 PIM3 PIM3 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PIP5K1A PIP5K1A PIP5K1-alpha, PIP5KIalpha, PtdIns(4)P-5-kinase 1 alpha ADP-Glo Lipid kinase Bi-weekly Lipid Kinase Panel Data sheet
PIP5K1C PIP5K1C PIP5K1-gamma, PIPKIg_v4 ADP-Glo Lipid kinase Bi-weekly Lipid Kinase Panel Data sheet
PKA PRKACA PKACa HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PKA (L206R) PRKACA (L206R) PKACa HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
PKA-DNAJB1 PRKACA-DNAJB1 PKACa, Hsp40, Sis1, RSPH16B HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
PKAcb PRKACB PKAcb, MGC41879, MGC9320, PKA c-beta HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PKAcg PRKACG PKAcg HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PKCa PRKCA PRKACA, PKc-alpha, PKCa, PKCalpha HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PKCb1 PRKCB (1) PRKCB1, PKCB, PRKCB2, MGC41878, PKC-beta, PKC-beta1, PKCb1, PKCbeta1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PKCb2 PRKCB (2) PRKCB1, PKCB, PRKCB2, MGC41878, PKC-beta, PKC-beta2, PKCb2, PKCbeta2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PKCd PRKCD MAY1, MGC49908, nPKC-delta, PKC-delta, PKCd, PKCdelta HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PKCepsilon PRKCE PKCE, nPKC-epsilon, PKC-epsilon HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PKCeta PRKCH PKC-L, PKCL, PRKCL, nPKC-eta HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PKCg PRKCG PKCC, PKCG, SCA14, MGC57564, PKC-gamma, PKCgamma HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PKCiota PRKCI PKCI, DXS1179E, MGC26534, nPKC-iota HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PKCmu/PRKD1 PRKD1 PKD1, PKD, PKCM, PKc-MU HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PKCnu/PRKD3 PRKD3 PKD3, EPK2, PKc-NU, PKD3, PRKCN HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PKCtheta PRKCQ PRKCT, nPKC-theta HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PKCzeta PRKCZ PKC2, PKCzeta HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PKD2 (G870E) PRKD2 (G870E) PKD2, HSPC187 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
PKD2/PRKD2 PRKD2 PKD2, HSPC187 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PKG1a PRKG1 (a) PKG1, PGK, PRKG1B, PRKGR1B HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PKG1b PRKG1 (b) PKG1, PGK, PRKG1B, PRKGR1B HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PKG2/PRKG2 PRKG2 PKG2, cGKII, PRKGR2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PKMYT1 PKMYT1 MYT1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PKMzeta PRKCZ (aa184-592) nPKC-zeta, PKC2, PKMzeta HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
PKN1-TECR (Tex1Pex10) PKN1-TECR DBK, PKN, PAK1, PRK1, PRKCL1, MGC46204, TECR-PKN1, PKN1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
PKN1/PRK1 PKN1 DBK, PKN, PAK1, PRK1, PRKCL1, MGC46204, PKN1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PKN2/PRK2 PKN2 PRK2, PRKCL2, PAK-2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PKN3/PRK3 PKN3 PRK3, PKNbeta, RP11-545E17.1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PLK1 PLK1 STPK13 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PLK2 PLK2 SNK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PLK3 PLK3 CNK, FNK, PRK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PLK4/SAK PLK4 SAK, STK18 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PRKX PRKX PKX1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
PYK2 PTK2B CADTK, CAKB, FADK2, FAK2, PKB, PTK, RAFTK, CAK beta HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
RAF1 RAF1 (Y340D/Y341D) c-RAF HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
RAF1 (R391W) RAF1 (R391W) c-RAF HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
RET RET CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
RET (A883F) RET (A883F) CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
RET (E732K) RET (E732K) CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
RET (E762Q) RET (E762Q) CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
RET (G691S) RET (G691S) CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
RET (G810C) RET (G810C) CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
RET (G810R) RET (G810R) CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
RET (G810S) RET (G810S) CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
RET (L730I) RET (L730I) CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
RET (L730M) RET (L730M) CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
RET (L790F) RET (L790F) CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
RET (M918T) RET (M918T) CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
RET (R749T) RET (R749T) CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
RET (R813Q) RET (R813Q) CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
RET (R912P) RET (R912P) CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
RET (S891A) RET (S891A) CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
RET (S904A) RET (S904A) CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
RET (S904F) RET (S904F) CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
RET (V738A) RET (V738A) CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
RET (V778I) RET (V778I) CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
RET (V804E) RET (V804E) CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
RET (V804L) RET (V804L) CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
RET (V804L)-KIF5B RET (V804L)-KIF5B CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, KIF5B-RET (V804L) HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
RET (V804M) RET (V804M) CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
RET (V804M)-KIF5B RET (V804M)-KIF5B CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, KIF5B-RET (V804M) HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
RET (Y791F) RET (Y791F) CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
RET (Y806C) RET (Y806C) CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
RET (Y806H) RET (Y806H) CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
RET (Y806N) RET (Y806N) CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
RET-BCR RET-BCR CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, BCR-RET HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
RET-CCDC6 (PTC1) RET-CCDC6 CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, CCDC6-RET HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
RET-KIF5B (Kex15Rex14) RET-KIF5B CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, KIF5B-RET HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
RET-NCOA4 (PTC3) RET-NCOA4 CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, NCOA4-RET HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
RET-PRKAR1A (PTC2) RET-PRKARA1A CDHF12, CDHR16, HSCR1, MEN2A, MEN2B, MTC1, PTC, RET51, PRKARA1A-RET HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
RIPK2 RIPK2 CARD3, CARDIAK, CCK, GIG30, RICK, RIP-2, RIP2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
RIPK3 RIPK3 RIP3, receptor interacting protein 3 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
RIPK4 RIPK4 Receptor interacting protein kinase 4, ANKK2, ANKRD3, DIK, MGC129992, MGC129993, PKK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
RIPK5 DSTYK SgK496, SHIK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
ROCK1 ROCK1 P160ROCK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
ROCK2 ROCK2 KIAA0619, ROC2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
RON/MST1R MST1R CD136, CDw136, PTK8, RON HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
ROS/ROS1 ROS1 ROS, MCF3 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
ROS1 (G2032R) ROS1 (G2032R) ROS, MCF3 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ROS1 (G2101A) ROS1 (G2101A) ROS, MCF3 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ROS1 (G2101C) ROS1 (G2101C) ROS, MCF3 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ROS1-GOPC ROS1-GOPC ROS, MCF3 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ROS1-TPM3 ROS1-TPM3 ROS, MCF3 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
RSK1 RPS6KA1 RSK1, HU-1, MAPKAPK1, p90Rsk HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
RSK2 RPS6KA3 RSK2, HU-3, MRX19, CLS HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
RSK2 (I416V) RPS6KA3 (I416V) RSK2, HU-3, MRX19, CLS HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
RSK2 (L608F) RPS6KA3 (L608F) RSK2, HU-3, MRX19, CLS HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
RSK3 RPS6KA2 RSK3, HU-2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
RSK4 RPS6KA6 RSK4 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
SBK1 SBK1 SH3-binding kinase 1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
SGK1 SGK1 SGK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
SGK2 SGK2 H-SGK2, dJ138B7.2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
SGK3/SGKL SGK3 CISK, SGK2, SGKL HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
SIK1 SIK1 SIK, MSK, SNF1LK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
SIK2 SIK2 QIK, SNF1LK2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
SIK3 SIK3 L19, QSK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
SLK/STK2 SLK KIAA0204, STK2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
SNARK/NUAK2 NUAK2 SNARK, DKFZp434J037 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
SNRK SNRK SNF1-related kinase HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
SPHK1 SPHK1 Sphingosine kinase 1 ADP-Glo Lipid kinase Bi-weekly Lipid Kinase Panel Data sheet
SPHK2 SPHK2 Sphingosine kinase 2 ADP-Glo Lipid kinase Bi-weekly Lipid Kinase Panel Data sheet
SRMS SRMS C20orf148, SRM, dJ697K14.1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
SRPK1 SRPK1 SFRSK1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
SRPK2 SRPK2 SFRSK2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
SSTK/TSSK6 TSSK6 FLJ24002, SSTK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
STK16 STK16 TSF1, PKL12, MPSK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
STK21/CIT CIT CRIK, STK21/CIT HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
STK22D/TSSK1 TSSK1B TSSK1, FKSG81, SPOGA4, STK22D HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
STK25/YSK1 STK25 YSK1, SOK1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
STK32b/YANK2 STK32B YANK2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
STK32c/YANK3 STK32C YANK3 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
STK33 STK33 STK33 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
STK38/NDR1 STK38 NDR1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
STK38L/NDR2 STK38L NDR2, KIAA0965 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
STK39/STLK3 STK39 STLK3, DCHT, SPAK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
SYK SYK SYK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
TAK1 MAP3K7 MAP3K7, TGF1a, MEKK7, TAK1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
TAOK1 TAOK1 TAO1, KIAA1361, MAP3K16, MARKK, HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
TAOK2/TAO1 TAOK2 KIAA0881, MAP3K17, PSK, PSK1, TAO1, TAO2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
TAOK3/JIK TAOK3 DPK, JIK, MAP3K18, TAO kinase 3 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
TBK1 TBK1 CDC37, HSPCA, HSPCB, IKBKG, NAK, T2K, TANK, TRAF2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
TEC TEC PSCTK4 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
TESK1 TESK1 TESK1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
TESK2 TESK2 TESK2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
TGFBR2 TGFBR2 HNPCC6, MFS2, RIIC, TGFbeta-RII, TBR-II, TRBII HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
TIE2 (A1124V) TEK (A1124V) VMCM, TIE-2, VMCM1, CD202B HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
TIE2 (P883A) TEK (P883A) VMCM, TIE-2, VMCM1, CD202B HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
TIE2 (R849W) TEK (R849W) VMCM, TIE-2, VMCM1, CD202B HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
TIE2 (Y1108F) TEK (Y1108F) VMCM, TIE-2, VMCM1, CD202B HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
TIE2 (Y897C) TEK (Y897C) VMCM, TIE-2, VMCM1, CD202B HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
TIE2 (Y897S) TEK (Y897S) VMCM, TIE-2, VMCM1, CD202B HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
TIE2/TEK TEK VMCM, TIE-2, VMCM1, CD202B HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
TLK1 TLK1 PKU-beta, KIAA0137 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
TLK2 TLK2 MGC44450, PKU-ALPHA HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
TNIK TNIK TRAF2 and NCK interacting kinase, KIAA0551, MAP4K7 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
TNK1 TNK1 TNK1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
TRKA NTRK1 MTC, TRK, TRK1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
TRKA (A608D) NTRK1 (A608D) MTC, TRK, TRK1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
TRKA (F589L) NTRK1 (F589L) MTC, TRK, TRK1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
TRKA (G595R) NTRK1 (G595R) MTC, TRK, TRK1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
TRKA (G595R/A608D) NTRK1 (G595R/A608D) MTC, TRK, TRK1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
TRKA (G595R/G667A) NTRK1 (G595R/G667A) MTC, TRK, TRK1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
TRKA (G595R/G667C) NTRK1 (G595R/G667C) MTC, TRK, TRK1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
TRKA (G595R/G667S) NTRK1 (G595R/G667S) MTC, TRK, TRK1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
TRKA (G595R/L657M) NTRK1 (G595R/L657M) MTC, TRK, TRK1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
TRKA (G667C) NTRK1 (G667C) MTC, TRK, TRK1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
TRKA (G667S) NTRK1 (G667S) MTC, TRK, TRK1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
TRKA (L657M) NTRK1 (L657M) MTC, TRK, TRK1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
TRKA-TFG NTRK1-TFG TRKA, TGF-NTRK1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
TRKA-TPM3 NTRK1-TPM3 TRKA, TPM3-NTRK1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
TRKA-TPR NTRK1-TPR TRKA, TPR-NTRK1 HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
TRKB NTRK2 GP145-TrkB HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
TRKC NTRK3 GP145-TrkC HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
TRKC (G623E) NTRK3 (G623E) GP145-TrkC HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
TRKC (G623R) NTRK3 (G623R) GP145-TrkC HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
TRKC (G623R/L686M) NTRK3 (G623R/L686M) GP145-TrkC HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
TRKC (G696A) NTRK3 (G696A) GP145-TrkC HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
TRKC (L686M) NTRK3 (L686M) GP145-TrkC HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
TRPM7/CHAK1 TRPM7 CHAK1 HotSpot™ Protein kinase Bi-weekly Atypical Panel Data sheet
TSSK2 TSSK2 DGS-G, SPOGA2, FLJ38613, TSK2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
TSSK3/STK22C TSSK3 STK22C, STK22D, SPOGA3 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
TTBK1 TTBK1 KIAA1855, BDTK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
TTBK2 TTBK2 KIAA0847 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
TTK* TTK ESK, MPS1L1, MPS1, PYT HotSpot™ Protein kinase Not included in any panel Data sheet
TXK TXK BTKL, PSCTK5, PTK4, RLK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
TYK1/LTK LTK TYK1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
TYK2 TYK2 JTK1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
TYRO3/SKY TYRO3 BYK, Brt, Dtk, Sky, Tif HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
ULK1 ULK1 UNC51, Unc51.1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
ULK2 ULK2 ATG1B, KIAA0623, Unc51.2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
ULK3 ULK3 FLJ90566, DKFZP434C131 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
VRK1 VRK1 VRK1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
VRK2 VRK2 VRK2 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
WEE1 WEE1 WEE1hu HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
WNK1 WNK1 KDP, KIAA0344, PHA2C, PRKWNK1 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
WNK2 WNK2 KIAA1760, NY-CO-43, P/OKcl.13, PRKWNK2, SDCCAG43 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
WNK3 WNK3 KIAA1566, PRKWNK3 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
YES/YES1 YES1 C-YES, HsT441, P61-YES, YES1, YES HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
YES1 (T348I) YES1 (T348I) C-YES, HsT441, P61-YES, YES1, YES HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
YSK4/MAP3K19 MAP3K19 M3K19, RCK, YSK4 HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
ZAK/MLTK MAP3K20 MLTK, mlklak, ZAK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
ZAP70 ZAP70 SRK, STD, TZK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
ZAP70 (Y319F) ZAP70 (Y319F) SRK, STD, TZK HotSpot™ Protein kinase Bi-weekly Mutant Panel Data sheet
ZIPK/DAPK3 DAPK3 ZIPK/DAPK3, ZIP, ZIPK HotSpot™ Protein kinase Bi-weekly Wild Type Panel Data sheet
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* Kinase targets are not part of the bi-monthly screening panels

Legend of HGNC References
Fusion: ALK-TFG; fusion protein including TFG and ALK
Complex: CDK4-CCND1; a complex of CDK4 and Cyclin D1 via coexpression
Mutant or deletion: FGFR3 (G687C); FGFR3 point mutant substitution Glycin 687 to Cysteine
Fragment: FAK aa411-686; FAK comprising amino acids 411 to 686. Indicated only when two different constructs are available.
CD: catalytic domain fragment
FL: full length
Isoforms: PRKCB (2); PRKCB isoform 2

 

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