CYP19A Inhibition Assay Service

CYP19A for compound screening and profiling assay using a fluorescence-based method to measure cytochrome P450 enzyme activity.

Target Overview
CAT#

CYP19A

Enzyme

Human CYP19A

Synonym

Aromatase, Cytochrome P450 19A1, Estrogen synthase, ARO1, CP19A

Scientific Information

P11511 (http://www.uniprot.org/uniprot/P11511)

Assay Properties
Substrate

Dibenzylfluorescein

Reaction

RH + O₂ + NADPH + H⁺ = ROH + H₂O + oxidized [NADPH—hemoprotein reductase]

Readout

Enzymatic activity

Reference Compound IC50s
Screening Location

Malvern, PA, USA

Further information

More information can be found on our website Cytochrome P450 Assay Services.

Reference compound IC50 for CYP19A