NSD2 SPR Assay Service

NSD2 for direct binding screening and profiling of test substance with surface plasmon resonance (SPR) technique.

Target Overview
Target

NSD2-SET

HGNC symbol

NSD2

Synonyms

Probable histone-lysine N-methyltransferase NSD2, Multiple myeloma SET domain-containing protein, Nuclear SET domain-containing protein 2, Protein trithorax-5, Wolf-Hirschhorn syndrome candidate 1 protein, WHSC1, KIAA1090, MMSET, TRX5

Scientific Information

O96028 (https://www.uniprot.org/uniprotkb/O96028/entry)

Screening location

Malvern, PA, USA

Further information

More information can be found on our website SPR Assay Services for Drug Discovery

Hit confirmation at 25 µM

Hit confirmation at 25 µM

The data were collected on a Biacore 8K using multi-cycle kinetics. The data were analyzed using a steady state affinity model.


Binding kinetics of SAM/SAH to NSD2-SET domain

Binding kinetics of SAM/SAH to NSD2-SET domain

The data were collected on a Biacore 8K using multi-cycle kinetics. The data were analyzed using a steady state affinity model.