Challenges in profiling and lead optimization of drug discovery for methyltransferases. Drug Discovery Today Technologies, 2015 by Andrew Khouri | Jul 6, 2023
Development and Use of Assay Conditions Suited to Screening for and Profiling of SET-Domain-Targeted Inhibitors of the MLL/SET1 Family of Lysine Methyltransferases. Assay and Drug Development Technologies, 2015 by Andrew Khouri | Jul 6, 2023
Screening and profiling assays for HDACs and sirtuins. Drug Discovery Today Technologies, 2015 by Andrew Khouri | Jul 6, 2023
A Highly Selective Dual Insulin Receptor (IR)/Insulin-like Growth Factor 1 Receptor (IGF-1R) Inhibitor Derived from an Extracellular Signal-regulated Kinase (ERK) Inhibitor. The Journal of Biological Chemistry, 2013 by Andrew Khouri | Jul 6, 2023